Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID76558 Canertinib GSE92742 MCF10A Human 6h 0.08uM EID0439
Types Number Response transcription factors
Up-regulation 73 TSC22D3; BMI1; TOB1; SMARCA2; NFIL3; MXI1; TFDP2; MECOM; TRIM16; SAP18; ZSCAN31; MEIS1; ATF3; ZNF165; HSF2; EDF1; HTATIP2; SUB1; CEBPA; ELF3; POU4F1; SIM2; CCDC59; ZBTB11; TRIP6; TMF1; HMGN3; OSR2; BTG1; MEOX1; CERS6; EZH2; REST; PBXIP1; YEATS4; ZNF467; SIAH2; MAF; MAFB; HOXA10; MED21; TBL1X; PIR; NR1H3; ELF1; FOXG1; KLF4; ZNF226; PHF8; HDAC1; NCOA1; AFF1; IRF7; TXNIP; CREG1; PSIP1; CITED2; CREB1; SATB1; LEF1; PAX6; NR1D2; AHR; TCEA2; TAF10; CREM; ATF5; FOXC1; NR2F2; PTTG1; TRPS1; TCFL5; HOXC6
Down-regulation 70 MYC; FOSL1; HMGA2; RBFOX2; ETV4; NANOG; SMAD7; ARNT2; NFATC1; HIC2; LIN28A; EGR4; ZIC3; FOS; NFATC4; ZFP36L2; EGR3; E2F3; ERG; BCL10; LZTS1; HOXA1; BHLHE40; POU5F1B; PHOX2B; GFI1; ZBED2; NFE2L3; EN1; FOXK2; DLX5; HOXB2; MYT1L; NFAT5; TGFB1; ATN1; LOXL2; ELK3; EPAS1; NFE2; ETV5; SNAI2; ERF; TSC22D1; HDAC9; HES1; NR4A1; MAGED1; TOX3; CTBP2; SATB2; YAP1; ZNF512B; FHL2; SOX10; SOX9; ERBB4; BCL11A; SMAD1; ARID5B; SMAD3; TLE1; ID1; MTF2; TFEC; ZMYM2; MTA1; STAT1; ZBTB20; TRIB3