Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID76555 Canertinib GSE92742 MCF10A Human 6h 10uM EID0439
Types Number Response transcription factors
Up-regulation 64 IKZF1; MNAT1; TSC22D3; HCFC2; XBP1; ID2; ARNTL; ING1; RBBP8; SAP18; NFIL3; SIX1; HMGN3; COPS5; RORA; SUB1; ITGB3BP; DNAJC1; MEOX1; IRF5; DDIT3; BMI1; BATF3; NFYC; EZH2; TBPL1; BRD2; CCDC59; TOB1; HOXC6; YEATS4; RNF141; TRIM29; HDAC6; CD3D; HMGB3; HOXA5; TRIP6; SIM2; TP53; ZNF226; HSBP1; RBL2; PSIP1; LITAF; MED24; SPIB; BRD8; JUP; ASCL1; TXNIP; BASP1; WT1; SMARCD3; PTTG1; NKX3-1; PLAGL1; CITED2; TFEC; NR1H2; ST18; RBPMS; LEF1; MYCBP
Down-regulation 106 MYC; FOSL1; EGR3; BCL10; EGR4; KLF10; ID4; TFAP2A; NPAT; TEAD1; ZNF551; ZNF232; TCF3; TCF20; DDX17; MGA; ZNF629; TAF1A; ZFP36L2; TRIM32; LZTS1; SIX3; ARNT2; ZNF117; ZFP36L1; THAP4; ZNF12; MEF2A; EYA2; SOX11; ZBED4; PCGF3; ERF; FOS; RBFOX2; ZNF43; NR2F6; CBX7; TFAP2C; E2F3; HIC2; ZNF112; FHL2; VEZF1; ZNF266; SMAD1; ZNF443; ZEB1; NEUROD1; FOXF2; ZBTB7A; ID1; EPAS1; MAFF; ARID1A; ZNF623; HMGA2; HDAC9; WWTR1; KAT6A; RREB1; SOX13; TEAD4; CDK9; MEIS2; ZNF512B; HOXB2; AHR; ERG; MXI1; ETS2; JUNB; ZFPM2; MNT; DLX5; EGR2; ZNF217; ETV5; ELK3; TCF7L2; E2F5; ENO1; SMAD3; CAMTA1; JUND; MED13; EYA1; SPEN; PHF20; ERBB4; HES1; PBX3; POU2AF1; ZBTB18; HOXD1; SSBP2; SCAND1; FOSL2; TLE1; ZBTB20; BHLHE41; MTA1; SMARCA1; STAT1; NFKB2; ZIC1