Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID74730 Azd-6482 GSE92742 MCF10A Human 24h 0.4uM EID0431
Types Number Response transcription factors
Up-regulation 212 ETV1; STAT5B; PCGF2; IRF3; PBX1; TGFB1I1; POU2AF1; FLNA; ZNF532; MAZ; GON4L; OLIG2; FOXO3; CBX4; ZNF580; CBFA2T2; NCOR1; CNOT6; ZNF444; ZBTB48; ZSCAN16; CEBPA; ZNF211; CREBL2; ZNF419; TAF6; SPEN; CHD3; HOXB13; IRF7; ZNF75D; NFATC4; RNF138; CALCOCO1; EN2; NR2F1; NANOG; KAT8; KAT2A; SRY; MAFB; ZBTB18; CREB3L1; SMARCC2; KLF4; ZNF606; MBD1; BNC2; SMARCA1; AHR; SOX13; ZNF692; SMAD7; RERE; SPIB; ARID1A; BACH2; CNOT3; ID4; ZEB1; PRDM4; UBTF; AEBP1; MYC; KAT2B; TRPS1; TRIM28; AES; NCOA6; RBFOX2; HMGA1; PBXIP1; NEUROD1; ZFHX3; ZNF263; ZNF7; FOXN3; DBP; IRF6; PRDM2; SETD2; TERF2; INSR; BRWD1; LOXL2; ZNF688; TRAK1; TCF4; PROX1; PTTG1; UBP1; SRCAP; TFAP2C; SMAD1; NRL; ARHGAP35; ETV6; BPTF; REPIN1; MGA; SLC2A4RG; RB1; BASP1; FOXE1; MBD2; ZNF423; FOXA1; TAF10; CLOCK; TEAD3; ZSCAN31; PAWR; ZNF83; MAML1; CTBP2; CARHSP1; ZNF623; GTF2I; CENPF; SIX1; CXXC1; PEG3; STAT2; BCL6; ETV5; WNT4; ARNTL2; ZSCAN18; BCL3; ZNF33B; JUND; TFCP2; PCBD1; ERBB4; MLLT10; TRIP11; ELF4; ZBTB14; ZNF512B; ZNF304; ATN1; LITAF; ZBTB1; NR0B2; NCOA2; GTF3A; SUPT6H; RUNX3; TRIM24; MEIS1; ZMIZ2; NPM1; ZNF652; KLF11; SMAD4; ZBTB20; NKX3-1; ZNF467; HLF; TLE2; SOX5; SMAD2; MECOM; MEIS2; MAF; FOXM1; TCF7; TRIM16; ZNF112; TCEA1; SMARCA2; SMARCD3; JUP; EED; IRF4; HOXB6; KDM4C; EYA2; PAX5; MYBL1; ELF1; SOX11; OSR2; NR3C2; ZNF24; FOSL2; DDX5; WWTR1; TBX3; RBPMS; TRIB3; SIAH2; GRHL2; ZNF264; IRF8; BCL11A; ZFPM2; PPARGC1A; BRD4; PRRX1; ASCL1; SNAI2; CD3D; SSX1; KLF10; TXNIP; ZNF274; IKBKAP; ZNF331; ARNT2; PBX3; TWIST1
Down-regulation 177 CDK7; HDAC2; CEBPB; NR2F6; DPF2; ENO1; ZNF562; PIAS1; DNMT1; MDFI; ZNF124; ARID3A; MED6; MSX1; ZNF335; SUZ12; FOXD1; BATF3; KMT2D; HMGN3; SMAD5; GMEB1; CTNNB1; SOHLH2; MDM4; CCNC; DNAJC1; TRIM32; SUB1; CREB5; SIM2; NR2C1; RBBP7; BTAF1; SKI; CTR9; FOXC1; TRIP6; YEATS4; RNF14; USP16; MAGED1; HOXB9; ETS2; EWSR1; THAP4; BANP; HOXA7; NFKB1; ZNF426; CCDC59; PLAGL1; MED4; CHD1; SAFB2; SERTAD2; HOXA3; HTATIP2; RFC1; MAFG; TOPORS; KAT5; BTF3; ADNP; ZNF14; CDC5L; ZBTB17; ELK1; HOXA1; ORC2; PIAS3; BLZF1; RORA; RELB; HSF2; BBX; ZNF205; HIVEP2; ZMYND8; HIC2; ZNF3; DDIT3; BMI1; SUMO1; HMGB1; ZBTB7A; ARNTL; THRA; PIR; PFDN5; TCEB2; ESRRG; TCEA2; RNF111; PCGF3; SSRP1; HEY2; SP3; TEAD1; POU2F2; TSG101; CNOT2; NFX1; RUNX1; COPS5; TAF12; ZNF468; PSMC3; EP300; E2F3; PHF8; ELF3; NFAT5; TRIM29; RFXANK; RNF141; ERG; MYT1L; ING3; PGR; TMF1; BAZ1A; UBE2B; DNMT3B; ZNF22; CCNE1; MDM2; TCF7L2; GATAD2A; ZNF222; CBX3; ZNF107; PRRX2; RXRA; CITED1; ZBED2; NRBF2; TAF9; MYRF; ID3; ILF2; TOB1; TGIF2; HMBOX1; CHD4; JUNB; HNRNPD; DACH1; PITX2; RCOR1; NFE2L2; SAP18; FOXL2; DLX2; ZBTB38; NR2F2; MYCN; CCNA2; TSC22D2; VPS72; EN1; YWHAB; SALL1; KLF5; GTF2A2; HDAC1; BRCA1; KLF2; KAT6B; EGR3; NUP62; STAT3; CITED2; ID1; TFEC; IFI16; KDM5B