Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID60664 Canertinib GSE92742 SKB Human 24h 10uM EID0342
Types Number Response transcription factors
Up-regulation 80 NR3C1; ATF5; TSC22D3; RXRG; LZTS1; NR5A2; NFIL3; DEK; CAPN15; PPARG; MXI1; MAFB; HIPK1; TRIB3; CBX6; SRY; RBPMS; DDIT3; FHL5; AHR; MKL2; HOXD1; TBX2; NRBF2; ASH2L; HOXD3; MITF; RBBP8; PROX1; IFI16; ATF4; ATF2; SIX3; SOX18; TWIST1; NFKBIA; TEAD1; BTG1; ALX1; BTF3; PBX3; CREM; UBE2B; ZEB1; HMGN3; TAF9; NKX2-1; ZNF232; PEX2; CREG1; KLF10; LPIN2; ISL1; ZNF516; ID4; TDP2; ZBTB16; KLF4; NFE2L2; ASCL1; MAF; ATF3; SOHLH2; MECOM; KAT6B; ZFPM2; GTF3A; PLAG1; SMAD6; SAP30; KLF9; ID1; TFAP2A; TBL1X; AFF1; NR1D2; NR2F6; POU2AF1; PEG3; CEBPD
Down-regulation 97 FHL2; MYCBP; SOX4; PUF60; CREB3L1; JUNB; TERF2; TBX21; ECD; UBE3A; DRAP1; ZNF562; SFMBT1; PPP1R13L; PAX5; SMARCD2; TFCP2; OLIG2; NCOR1; TAF1D; LOXL2; RNF141; RBBP7; POU2F1; POU4F1; ZNF184; USP16; ARID1A; TCF3; BRCA1; SMAD3; NR2F2; MED23; CRYM; EZH2; REL; NFATC3; IRF9; NEDD8; AES; EGR1; CBFB; CREBZF; ETV4; ZNF85; ZNF45; PLAGL1; AR; ZNF432; TFEB; MYB; RORA; FOXJ2; MAGED1; MYRF; HDAC9; HOXC10; MEF2C; SUV39H1; CCNA2; SAP18; IRF8; TLE1; IKBKAP; JUP; HMGB2; IRF6; TCF7; SMAD1; MEF2A; EHF; TLE4; LMCD1; TCF4; SUB1; ZNF443; SIAH2; BCLAF1; NCOA1; SIM2; MYBL1; SLC2A4RG; NKX2-2; SCAND1; BCL11A; APEX1; ZBTB18; FOXM1; TRIP6; SOX9; CITED2; FOXC1; ERG; ZNF274; KDM5D; GATA2; LEF1