Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID58711 Canertinib GSE92742 HA1E Human 6h 10uM EID0328
Types Number Response transcription factors
Up-regulation 59 FOXO4; XBP1; ST18; SETDB1; RAD21; ERBB4; ZMYM2; ATF4; CDK7; TOX; DDIT3; CEBPB; TSC22D3; RB1; CEBPD; ASCL1; TCEA1; CALR; GTF3A; CD3D; MYCN; TERF1; IRF8; HBP1; BRD8; NR1D2; SMAD5; ZNF331; HIVEP2; RBPMS; SAP30; ZNF24; ACTL6A; CBFA2T3; MTF2; DBP; EMX2; NEUROD1; HTATIP2; PNRC1; BCL11A; FOS; UBE2B; CITED2; PAX6; REPIN1; MED1; JUP; MNDA; RFX5; RBBP8; TRPS1; HMGB2; TRIM22; TOX3; TP53; MXI1; INSM1; PEG3
Down-regulation 69 FOSL1; JUN; NFKBIA; MYC; KLF6; SFPQ; USP22; FHL2; LOXL2; NR2F6; MAFF; DLX2; PDLIM1; CTBP2; KLF10; CRK; LITAF; RELB; ID1; TGFB1I1; HOXB6; ELK3; PPRC1; E2F3; HOXD11; MAGED1; ZBTB18; ZNF593; FLNA; SMAD3; HMGA2; ATF3; EGR2; MECOM; TEAD4; HOXB5; TCF12; CHD4; ETS2; ARID5B; PRRX1; ID3; TCF7L2; ETV4; STAT4; WWTR1; NKX3-1; NR4A1; HHEX; KLF2; TGFB1; VEZF1; NR2F2; HOXB7; ZFP36L1; MEIS2; ZNF512B; HOXB2; SMARCA1; TBL1X; MYRF; EYA2; ATF5; ESR1; HOXA11; PTRF; TFAP2A; IKZF1; HOXA5