Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID18340 Canertinib GSE70138 MCF10A Human 3h 0.37uM EID0024
Types Number Response transcription factors
Up-regulation 53 TSC22D3; JUN; ID2; MEIS2; ZNF423; MEIS1; HIVEP1; HLX; MEOX2; PLAGL1; ISL1; ZFHX3; CUX2; EYA1; SOX13; TCF21; SMAD6; ID3; TCEA1; MED14; TOX; HMGN3; FOXF1; FOXN3; OSR2; HMGB2; AR; SATB1; NR3C2; PHIP; ESRRG; RARG; TBX2; PBX3; TCF7L1; TLE4; LEF1; SOX17; FOXF2; WT1; TWIST1; ZFPM2; GATA6; MECOM; MYCL; ZNF331; BHLHE40; SNAI2; TLE1; ZBTB20; DACH1; ATF3; ID1
Down-regulation 38 CRK; FOSL1; MYC; HMGA2; FHL2; HOXA5; NRIP1; HES1; GATAD2A; EGR1; ZKSCAN1; CREB5; MAFG; MAFF; MED13; NR2F6; BAZ1A; BCL10; KLF10; HOXC10; FOXC1; HHEX; HMGA1; ZNF430; EGR3; ADRB2; SMARCA1; SOX9; HOXB6; HOXC6; ZBTB38; ELK3; HOXB2; IRX5; TOX3; FOS; KDM5D; IKZF1