Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID18339 Canertinib GSE70138 MCF10A Human 3h 1.11uM EID0024
Types Number Response transcription factors
Up-regulation 47 TSC22D3; PAX6; ID2; FOXN3; PIAS1; FOXO4; FOXM1; ZNF32; BNC2; PBX1; NHLH2; ZMYND8; HMBOX1; ZNF304; KAT6B; ZMIZ1; PLAGL1; GLI2; TCF4; AEBP1; HMGB2; HEY1; CEBPG; MXI1; EMX2; SMAD6; PHIP; EHF; NFATC3; MEIS2; ID3; TRIM22; NR1D2; KAT2B; KDM5D; ZNF302; ZBTB16; BTG1; PEG3; PBX3; MAF; ELF5; INSM1; SATB1; ZBTB20; MEIS1; TLE1
Down-regulation 43 FOSL1; MYC; HMGA2; FHL2; NRIP1; HES1; SMAD3; TRIM32; KLF10; EGR1; EGR3; E2F6; AGO2; NPAS2; BHLHE40; ETV4; ADRB2; ETV5; TRIM16; JUN; ELK3; IRF2; FOXA2; SOX9; RUNX1; STAT3; MEOX1; NFE2; ESR1; EGR2; MAFF; FOXC1; HMGA1; ETS2; CBFB; IRF4; ZFP36L2; MEOX2; HOXB2; MYB; BASP1; BHLHE41; IKZF1