Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID18109 Canertinib GSE70138 MCF10A Human 3h 3.33uM EID0023
Types Number Response transcription factors
Up-regulation 38 TSC22D3; FOXO4; XBP1; MITF; RBBP8; ADNP2; SMAD4; DDIT3; HMGB2; E2F2; ATF4; NR1H2; SMARCA2; SMARCA4; TXNIP; EMX2; TRIM29; TBL1X; CITED2; JUND; RBPMS; SIAH2; FOSL2; KLF11; JAK2; ISL1; HLTF; ZBTB20; PEG3; ZSCAN18; MAFB; HOXA5; KLF4; ZNF331; ZFPM2; PIR; ZNF91; NR2F6
Down-regulation 30 FOSL1; MYC; HMGA2; ETV1; ADRB2; E2F5; SIX2; RUNX3; EGR1; FHL2; EGR3; ZNF267; EGR2; ZFP36L1; SMAD3; ERG; SOX9; CHD7; ETS2; FOXO1; TLE1; MYBL1; CTBP2; NKX2-1; KLF10; IFI16; ELK3; ASCL1; BASP1; NR4A2