Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID18108 Canertinib GSE70138 MCF10A Human 3h 10uM EID0023
Types Number Response transcription factors
Up-regulation 226 GATA2; PEG3; NFE2; FLI1; CEBPA; CBL; ARID3A; SOX4; ARRB1; MYCN; E2F2; NR3C2; ZIM2; PROX1; CIITA; SOX5; GATA4; ZNF177; ZNF552; SHOX; ZNF675; SIX6; THRA; ZNF710; RORB; ZNF665; ZKSCAN8; FOXL2; HIPK3; TGIF1; EPAS1; SSX7; ZNF208; ZNF415; KLF3; DLX2; BRDT; ZNF423; TULP2; TAL1; SKI; ZNF816; RBPJ; CBX6; ZNF467; ERBB4; SPI1; ZNF471; SMARCA1; KAT6B; TOX; ZFP2; SOHLH2; GBX2; RING1; ZNF835; HOXA2; POU4F2; CBX4; ZNF74; ZNF253; ZNF132; NFIX; ESRRG; ZNF331; ZNF528; TRIM24; PRDM13; ZNF141; GLI2; ZNF492; ID4; ZNF334; PRDM1; ZNF780B; JAK2; ZNF682; RFX3; SOX18; ASCL3; SUPT3H; ZNF225; CDIP1; TLX3; NCOA1; ZNF175; ARID3B; SCAI; NEUROD2; RXRA; MAML3; ZSCAN18; TP73; CARF; CD3D; ZFPM2; PROP1; ZNF10; PAX5; MEF2C; NR5A2; HINFP; TSHZ2; TBX1; FOXN3; ZNF232; TRPS1; ID3; THRB; ZNF117; ZNF695; FEZF2; ZNF257; INSR; DCC; ZNF43; HBP1; PRDM14; LMCD1; ZKSCAN1; ZNF711; MDM4; TTF2; PHIP; CREM; CBFA2T3; HEY1; HIF3A; EN1; HHEX; NR2F1; KLF4; EMX1; BACH1; SOX2; HDAC5; PAWR; HIC2; HEY2; TFDP2; TCF7L2; PRRX1; VGLL1; BARX1; SSX1; ZNF124; HIPK2; RARG; KLF11; ZNF154; TLE4; ZSCAN31; ZNF273; SMAD6; MECOM; SPDEF; ZNF165; CREB3L2; FOXF2; AEBP1; LHX3; HLX; ZMIZ1; NHLH1; TCF7L1; ZNF85; IRF6; ATOH1; NFATC4; ISL1; PRDM12; BCL11A; WWTR1; ZNF93; PBX3; NR4A2; ZNF345; ARID5B; ZIC3; ZNF623; NR1H4; ZNF573; HDAC9; TFEC; SOX3; POU2AF1; CAMTA1; ZNF589; NR1H2; GATA6; TCF4; CUX2; ETS1; PNRC1; EMX2; VDR; WT1; FOXF1; TCF21; NR4A3; SALL2; OSR2; NANOG; MEIS2; LEF1; MNDA; ZEB1; ZBED2; NEUROD1; LIN28A; PAX6; JUP; ZNF512B; ST18; MEIS1; TBX3; MAF; SNAI2; IRF8; SOX17; IRF9; ZNF91; NFATC3; VPS72; TRIB3; NR2F6
Down-regulation 47 MYC; FOSL1; CREG1; NRIP1; NFKBIA; HOXA10; ADRB2; RNF6; COPS2; HES1; CRY1; ARID4B; ENO1; SFPQ; TSC22D2; HNRNPD; USF2; ZNF267; FHL2; NCOA4; ZMIZ2; TRIM28; PRKDC; IKBKAP; AFF1; ATF1; ELF1; HOXB7; TP53; CTR9; MITF; EGR1; MTDH; GTF3A; HOXC6; SPEN; BHLHE40; CHD7; DNAJC1; TRIM16; BMI1; MAGED1; HDAC1; NR2F2; HOXA5; PUF60; KDM5D