Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17880 Canertinib GSE70138 MCF10A Human 3h 0.04uM EID0022
Types Number Response transcription factors
Up-regulation 116 HES1; EGR1; ZFHX4; TSC22D3; ID2; FOXG1; NR2E1; NR1I3; TAF9B; KDM5B; PNRC1; HIPK2; SMAD4; THAP10; PAX6; RORA; PBXIP1; ING4; HAND1; ZMIZ1; KLF13; PIAS2; RBPMS; PHOX2B; HOXC4; TWIST1; ARNTL; HBP1; FOXN3; PROX1; PRDM14; TRIM29; ZNF835; CALCOCO1; ATF3; MAFB; MECOM; BCL6; ZNF711; CREBL2; DACH1; ZNF75D; SRY; RORC; ISL1; SOHLH2; SMAD6; SATB1; TFEC; BHLHE40; ZNF532; CRYM; SSBP3; BHLHE41; MYRF; AES; ZNF423; MEIS1; TLE4; SOX13; PRRX1; TCF4; SHOX2; THRA; ZNF175; EYA1; BRD7; EN1; NR5A2; RBL2; MYCN; MEIS2; TBX3; BTG1; CNOT2; AHR; PPP1R13L; KLF5; WNT4; ZNF467; CREM; CERS4; KAT2B; TRPS1; NR4A1; HOXD1; VPS72; PFDN5; TP63; FOXF2; TRIM22; IRF6; HEY1; SIX3; HOXB2; SOX4; INSM1; SPDEF; SCAND1; NFATC4; SNAI2; TXNIP; HOXC6; CREB1; TOX; BCL11A; DLX5; KLF11; HOXB6; TCF7L2; SOX17; IRF8; FOSB; PITX1; ESR1; ID4
Down-regulation 46 FOSL1; MYC; FHL2; HMGA2; CHD7; NELFB; ATF1; SIX1; CDK8; BCL10; ZBTB11; SP140L; SF1; CCNE1; ZZZ3; DEAF1; HNRNPD; YAP1; ADRB2; SMAD3; CBFB; BACH2; AFF1; PBX3; GATAD2A; TSC22D2; SREBF1; JUNB; ETV1; BMI1; CRY1; ELK3; PDLIM1; EYA2; PRKDC; NRIP1; SMARCA5; LITAF; BAZ1A; MYB; CRK; EED; MAGED1; FLNA; FOXJ3; NR4A2