Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17877 Canertinib GSE70138 MCF10A Human 3h 1.11uM EID0022
Types Number Response transcription factors
Up-regulation 37 TSC22D3; DAXX; KDM5D; IRF7; ZMIZ1; RXRA; ARID5B; RORA; SLC2A4RG; TFEC; PCGF2; ID2; TWIST1; WT1; TRIM22; EMX2; HMGN3; ZNF43; ZNF423; BCL6; PSIP1; TRIM29; BNC2; ZNF512B; MAGED1; MYB; JUND; MYBL1; BTG1; ZNF117; MEIS1; TRIP6; ZSCAN18; FOXJ3; JUP; ESR1; MEIS2
Down-regulation 36 FOSL1; MYC; HMGA2; FHL2; EGR1; HES1; MAFF; JUNB; TSC22D2; MLXIP; ING3; CHD7; EGR3; EGR2; TGFB1I1; ADRB2; ZBED2; CREG1; ETS2; SMAD3; DLX2; CCNE1; CALR; NPAS2; PURA; FOSB; ASCL1; NKX2-2; NR4A2; NR4A1; PDLIM1; MED1; SATB2; SMARCA1; KLF4; SATB1