Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17650 Canertinib GSE70138 MCF10A Human 24h 0.12uM EID0021
Types Number Response transcription factors
Up-regulation 374 HDAC6; TSC22D3; PNRC1; HBP1; ZSCAN31; ZNF33B; SRCAP; WNT4; BTG1; MYCN; HEY1; MEIS1; ZNF136; ZNF764; ZNF629; OSR2; CREG1; SSX3; FOXO3; ARNT; CALCOCO1; MEOX1; ZKSCAN4; ZNF606; ZNF350; SSBP3; GATA3; IRF9; ZNF91; ZNF652; ZNF768; ZNF264; NFE2L2; ELF4; SP1; MYCL; ZNF224; CUX1; SUPT7L; ZNF467; HMBOX1; PKNOX1; CDX2; IRF6; ZBTB43; CARF; ZNF257; ZFP2; ZKSCAN8; ZBTB39; BAZ2A; TCF25; SETDB1; CREBL2; PBXIP1; ZNF14; ZNF174; ZNF536; TFEB; CBX4; JUNB; MNDA; RBL2; COPS2; CIR1; ZNF12; FOXF1; ZKSCAN3; ZNF688; SOX12; ZKSCAN1; HNF4G; HIC2; PHF1; NHLH1; FOXA2; HR; MYF5; TBX10; MYRF; ZNF254; RFX7; MYOG; SREBF2; RING1; RORC; ZNF711; TRIM29; ZSCAN2; ZNF354A; NHLH2; MZF1; ZNF93; ZBTB3; ZNF124; DYRK1B; EYA3; ING4; ZNF44; TAF1C; SPI1; REL; KDM4A; ZBTB44; ZSCAN18; ZNF816; ZNF345; ZBED1; ZNF669; FOXO4; HIF3A; HESX1; LMO1; ZNF141; GTF2I; ZNF223; PAX2; TCF7L2; ZNF217; LMX1B; HINFP; THRB; TAF5L; TRIM24; ATOH1; ZNF573; EPAS1; DLX4; TULP1; HIVEP1; ZNF510; FOXJ2; SALL1; SOHLH2; FOXN2; NR6A1; SALL2; ZNF140; ZNF492; ZNF221; ZNF512B; ZNF253; TP63; ZNF8; ZNF155; ATF3; KAT2B; ZNF208; CBX7; HOXA4; ZNF415; TFEC; ZNF550; MAZ; ZNF358; ZNF85; ATN1; MAML3; FOXN3; ZNF506; MNT; BAZ2B; OLIG2; TBX4; TEAD3; POU2F1; NCOR2; GLI2; SSX1; ZNF225; NR1I3; ZNF362; ZNF423; ZIC3; BRWD1; MDM4; KLF13; IRF8; ONECUT1; ZNF175; ZNF551; ZNF117; ZNF665; SSX7; ADRB2; HDAC9; RFX2; BNC1; BCL6; PRDM1; CBFA2T3; CEBPD; LMCD1; ID2; KLF3; CIC; TXNIP; SSBP2; ZNF43; GATA6; DACH1; ARID5A; ZNF177; SNAI2; SMARCD2; AFF2; CREBZF; ZSCAN9; ZNF135; ARID1A; MECP2; L3MBTL1; BCL11A; ZNF112; ERBB4; GATA1; KDM5C; ZNF268; ZNF675; HOXB13; TRIM16; IRX4; NFE2L1; TSC22D1; BRD4; KLF1; PHIP; CDIP1; REPIN1; MXI1; ZNF770; SMAD6; ERF; ZNF500; ZHX2; PKNOX2; ZNF75D; BRD2; TSHZ2; EMX1; ZBTB16; PHOX2B; FOXH1; YBX2; POU4F2; SMARCC2; ZNF682; MXD4; MKL1; RXRA; PPP1R13L; ZNF160; TFAP2A; MBD4; GFI1B; SPIB; CHD9; IRF1; KLF4; AES; CCNT1; PRDM14; SP4; NR1H4; BCL3; TULP3; ZKSCAN7; CHD2; CREB5; EN1; SCAI; MEIS2; ZNF248; ZNF544; ZNF329; CERS4; CIITA; NFATC4; MYT1; NR3C2; BARX1; ZNF189; ERBB2; ID3; CUX2; E2F5; BACH1; PAX6; HTATIP2; VENTX; FOXF2; JAK2; HLX; NCOA3; NEUROD1; SOX18; NR1H3; VPS72; SOX3; CSDC2; ZFP36L2; DDX17; ZNF611; TP53; ZIC1; MITF; TAL1; PRDM2; ZNF219; POU2AF1; RARG; TLE2; INSR; NR5A2; NCOA2; CRYM; RSF1; PEX14; PRDM12; HOXB5; DAXX; LIN28A; ZNF195; SHOX2; TOX3; ELF3; JUP; TCF7; ESRRG; NFATC1; NFAT5; ARID5B; NFKBIA; KLF9; RFX5; CEBPA; HOXD1; MED13; TCEA2; INSM1; VGLL1; TRPS1; SIX3; LOXL2; TCF21; ARNT2; SOX13; TFAP2C; MAFB; DLX5; TCF4; MEOX2; EHF; KLF5; PIR; KLF11; RORA; DLX2; FOSL2; NFE2L3; TRIM22; ID1; MAF; TRIB3; TOB1; TLE1; SOX17; ZFPM2; E2F2; BHLHE41; PBX3; MECOM; IKZF1; MEF2C
Down-regulation 104 FOSL1; CCNA2; HMGA2; EZH2; TCERG1; RUVBL2; PARP1; DRAP1; RBM14; PSMC3IP; PTTG1; BRCA1; TRIM28; YWHAB; FHL2; DR1; MYCBP; HMGB2; HMGB1; GTF2A2; NUP62; PDLIM1; HNRNPD; RBBP8; RUVBL1; CHAF1B; CDK2; SUZ12; HDAC2; ITGB3BP; BCLAF1; BATF3; CTR9; TFDP1; SMARCA5; NFIB; EGR3; RBL1; CENPF; SSRP1; WHSC1; EYA2; RBM39; WDR77; VEZF1; EGR4; SMARCA1; POU4F1; ETS1; RBBP4; SAP30; EGR1; NCOR1; WWTR1; KLF6; ZNF281; FOXM1; MED24; BAZ1A; PTRF; DEK; CEBPG; PA2G4; PRKDC; ATF4; NPM1; ATF5; RELA; CCNC; UBE2I; RAN; ZNF146; PUF60; NEDD8; PITX1; FOXK2; URI1; MLXIP; ENO1; HLTF; EGR2; COPS5; YBX1; SFPQ; SUV39H1; CBFB; MSX1; HMGA1; PSIP1; XBP1; BHLHE40; IFI16; MYBL2; MYB; HHEX; PEG3; ZBED2; TBL1X; RBPMS; SOX9; CITED2; AFF1; HOXC6; ELK3