Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17649 Canertinib GSE70138 MCF10A Human 24h 0.37uM EID0021
Types Number Response transcription factors
Up-regulation 633 TSC22D3; HINFP; ERBB4; ZNF669; EZH1; CALCOCO1; HOXC8; IRF9; ZNF253; ZNF816; NHLH1; ZNF350; CBX4; WNT4; CREG1; ZBTB43; ZNF44; ZNF93; HBP1; ZSCAN32; ZKSCAN4; NRL; ZNF222; RING1; THRB; ASCL3; ZNF688; PNRC1; ZNF76; ZNF430; KLF13; KAT2B; ZNF91; SRCAP; ESRRB; ZNF136; TUB; ZNF606; NEUROD2; GATA3; MEIS2; GBX1; ZHX2; RARB; ZKSCAN3; ZNF665; ALX3; FOXN1; ING4; AFF2; CRYM; LHX3; FOXJ1; ZNF611; PRDM2; ZNF506; FOXH1; ZNF778; DBP; CBFA2T2; ZNF467; ZSCAN16; HOXB5; NEUROG1; ZNF154; TULP1; NFATC3; ZBTB44; NFE2L2; HDAC9; ZNF274; PRDM1; ZNF586; TBX21; EPAS1; ZKSCAN8; THAP3; TULP2; PLAG1; ZNF667; VENTX; PROP1; ZNF74; SOX21; THRA; NFKB2; BCL11A; CRTC1; OSR2; FOXP3; LMO1; ZXDC; ZNF8; SOX5; NFATC4; SCRT1; SALL1; BNC2; GLI2; ZNF552; PITX3; ETV3; NR5A1; HDAC11; MED31; ZNF235; NEUROG3; IFNB1; ZNF415; TAF11; CDX4; ZNF573; ZSCAN9; FOXE3; ZNF394; SIRT2; ZNF175; TEAD3; ZNF85; NR1I3; RBPJL; PRDM14; ZNF132; MYRF; CSDC2; ZNF197; DLX5; TBX5; RARG; TFDP2; THAP7; ATOH1; ZNF419; SIM1; ZNF140; TLX3; ZNF221; HOXB1; HOXC11; ZNF423; MAP3K10; FOXF2; TP63; HEYL; SOX17; GLI1; ESR2; HSF4; EYA3; ZIC1; EMX1; KLF15; RFX3; CBFA2T3; NEUROD1; ZNF264; ZIC4; SSX7; CEBPD; TFDP3; SIX5; ZNF550; ZBTB7B; FOXL1; ZNF391; ZNF589; TBX10; ETV2; TBR1; DCC; NR0B2; NEUROD4; ZNF510; SCAI; ACTL6B; ZSCAN2; CRX; SUPT7L; SOX2; ZNF268; TRIM24; ZFP2; ZIC3; CCNH; ARID5B; RXRG; HESX1; SHOX; POU6F2; NR2C2; ZNF426; ZNF711; NR1H4; ZNF343; ZNF276; ZNF304; PBXIP1; CHD2; VAX2; ZNF345; KLF11; ZNF682; DYRK1B; TSHZ2; TAF6L; NR1H2; RAX; HOXA6; ATF3; BARX1; SOX3; ZFPM2; EN2; MECP2; HNF4G; CBX2; ZNF695; GCM1; TBX1; ZNF571; HOXA4; SRY; SETDB1; BNC1; ZNF671; RORC; RFX1; PRDM12; TBX6; GATA1; TBX4; ZFHX2; EVX1; ATF7; ZNF134; ZNF225; SUPT3H; POU2F3; HOXB8; EP300; ZNF75D; CIITA; ZBTB7C; POU6F1; ZNF223; AIRE; NKX6-1; PKNOX2; ZNF160; TULP3; ESRRG; TEF; APBB1; ZNF507; ZNF224; LZTR1; CBX7; ZNF250; SALL2; ZSCAN18; BCL6; ZNF257; IKZF4; CUX2; VGLL1; BHLHE40; NOCT; ZNF329; ZNF771; TCEA2; PAX6; ZNF770; HAND2; MAML3; TRIM29; NEUROD6; RFXANK; MYOG; ZFP30; HOXA2; MZF1; CDIP1; NHLH2; ZNF442; GFI1B; LHX2; TP73; ALX4; GRIP1; POU3F3; ID4; PHF1; PDX1; POU5F1B; ZNF749; ZNF234; ZNF180; ZNF43; ARNT; DDIT3; FOXN3; FOXD3; NFE2; ZNF701; TLX1; NFIX; VPS72; ZNF529; ZKSCAN7; STAT2; TBX3; ZNF471; GBX2; FOXE1; ZNF556; DLX6; RFX2; CBL; KLF3; MXI1; SSBP3; ZNF211; ZNF835; ZNF500; ZNF768; PIAS1; HOXD12; ONECUT1; ATF2; KDM5C; PAX7; IKZF3; ETV6; NR6A1; HIC2; FEZF2; TAF4B; SOX14; ZNF446; PAX3; POU4F3; PRDM16; SOHLH2; ZNF549; SNAI1; CIR1; TWIST1; NEUROG2; ZFP37; TFEB; ATF6B; SP1; LYL1; BACH2; PPARA; ZNF14; ONECUT2; BPTF; PRDM5; PRDM10; POLR3C; LMX1B; GSC2; ZNF34; HMBOX1; REL; BTG1; ZNF33B; GATA4; ZNF266; TFAP2A; ZNF480; PAX1; ZNF623; TBX19; FHL5; ZNF174; ZNF254; ZNF780B; POU2F1; SOX18; ZNF10; ZBTB16; LHX1; JAK2; MEIS1; NR4A3; MAPK8IP1; HOXB13; ZIM2; VHL; PIAS4; TBL1Y; SNAPC4; ZNF81; MYCL; SHOX2; SP140L; TERF2; FEV; ZNF362; ZSCAN31; FOXF1; ZXDB; TCF4; MED25; LIN28A; DLX2; DOT1L; NPAS1; NR5A2; ZNF215; KLF8; ARL2BP; RORB; ZKSCAN1; ZNF551; ZNF536; ZNF444; ZNF79; NFE2L3; MYF5; GCM2; ZNF334; HIF3A; LBX1; ZEB1; ZNF814; HNF1B; PRDM9; HEY1; DLX4; ARID3B; ZNF157; WHSC1L1; PEX14; SIX3; ZNF165; ZNF214; ZNF117; MBD1; SUMO1; YEATS2; OVOL2; ZNF654; ZNF674; ZNF492; INSM1; ARID3A; ZBTB39; PAX4; ZNF80; E4F1; NCOA3; SKIL; ZNF141; SP2; TRIM22; KLF1; NFIC; UTF1; HOXC5; TCF7; FOXI1; MYCN; STAT4; TLX2; KDM4C; AFF3; ZBTB3; SP4; NAB2; FOSL2; ZNF112; TGIF2; GON4L; FOXA2; ZNF407; HNF4A; ZNF493; HOXA3; FOXO3; PCGF3; KLF7; TAF1C; MAK; RSF1; TCF21; ZFHX3; TAF1; BANP; PFDN5; CD3D; CREB3; KMT2D; BRDT; ZNF135; POU2F2; TOX; SOX13; FOXB1; ZNF219; SNAI2; ZNF440; FOXJ2; HOXA11; FOXL2; BRD4; IRF6; BRWD1; ZNF217; CUX1; ZNF354A; ARID5A; DMRT1; IRF8; SUPT4H1; ST18; HLX; TCF3; OVOL1; RXRA; SOX1; MED17; PBX3; MLLT1; ZNF443; NCOA2; ZNF331; ZNF675; ZNF468; IRF1; ZBTB20; CARF; TXNIP; JUNB; POU1F1; HIRA; GFI1; CERS4; GRHL2; FOXO1; HEY2; TRIB3; TRPS1; HOXD1; BACH1; MXD4; HDAC5; MYT1L; E2F8; JUND; HIVEP1; IRX4; SMARCA1; AR; SPDEF; MEOX2; ISL1; MECOM; ZNF12; PAX5; ELF4; TADA3; ZBTB17; CAMTA2; LMCD1; ZNF358; PHIP; TAL1; GATA2; ZNF512B; NR4A1; RUNX1; IL16; FOXG1; DACH1; IFI16; ZNF562; NR4A2; ZNF148; BHLHE41; PEG3; POU2AF1; HIPK2; PAX8; EYA1; JUN; ZNF239; ZFP36L2; MNDA; HAND1; NFATC1; NR1D2; ZNF232; SPIB; AEBP1; ZNF652; CITED1; ID1; BRD2; SMAD6; DAXX; SCAND1; PBX1; LEF1; ATN1; ZNF721; RORA; SOX10; GATA6; KLF9; SMAD1; TLE2; WT1; MAF; HOXB6; SSBP2; EHF; MEF2C; HOXB2; HHEX; NANOG; TLE4; ARNT2; INSR; ESR1; IKZF1; SOX11; E2F2; SATB1; EMX2; TFAP2C
Down-regulation 118 FOSL1; CCNA2; TFDP1; TCERG1; EZH2; FHL2; PARP1; MYCBP; C1QBP; USP22; RBM14; DRAP1; BAZ1A; TRIM28; GTF2A2; YBX1; HMGA2; PTTG1; ITGB3BP; NPM1; NUP62; HSF2; MAGED1; SUB1; RUVBL2; CBFB; PPRC1; CENPF; UBE2I; MYC; RHOA; ENO1; BCLAF1; RBBP4; EGR1; RAN; HMGA1; DR1; HMGB1; SSRP1; FOXJ3; ABL1; SMARCA5; PA2G4; YWHAB; TAF10; SFPQ; RBL1; HDAC2; BRCA1; CTR9; NCOA4; BMI1; EDF1; SNW1; BRD8; ASH2L; CBX5; PSMC3IP; SND1; TBL1XR1; ATF1; DNAJC2; PSIP1; HOXC6; EED; ETS2; HOXB7; TAF1D; AFF1; TRIM32; SF1; PITX1; RCOR1; PURA; CTNNB1; SMARCC1; KAT7; JARID2; WHSC1; MTDH; SMARCE1; XBP1; CALR; SUV39H1; NFIB; HLTF; CRY1; HMGB2; FOXM1; MBD2; HMGB3; SAP30; BAZ1B; NRIP1; FOXD1; NR2F2; ELK3; CNOT1; WWTR1; HNRNPD; MAX; RNF6; PCGF2; BATF3; FLNA; SMAD2; BRD3; TCFL5; TSC22D2; NFKB1; IKBKAP; HOXC10; DEK; SMARCA2; SOX9; ELF1; PUF60