Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17646 Canertinib GSE70138 MCF10A Human 24h 10uM EID0021
Types Number Response transcription factors
Up-regulation 380 TSC22D3; PEG3; CALCOCO1; FOXO4; BTG1; TFDP2; SP2; ZNF426; CIITA; PNRC1; PBXIP1; HBP1; EP300; TBX6; SUPT7L; HIPK1; WNT4; KAT2B; ZNF91; MEOX1; HDAC5; SP100; SP140L; EZH1; ZIC4; ZSCAN2; ZNF136; MZF1; ZNF135; BPTF; FOXJ1; ZNF224; FOXP3; ZNF688; ZNF131; IRF9; ZNF430; ZSCAN16; GBX2; TBX21; ZNF14; ZNF764; CIR1; ASCL3; PRDM2; ARID5A; ELF4; GTF2F1; CSDC2; NR3C2; KDM5D; CDX1; CD3D; ZNF557; HOXB1; CREBL2; ARNT; PAX1; NR5A1; OSR2; HOXB3; ZNF44; TLX1; IKZF1; MED23; ALX3; TAF11; ZBTB43; ZNF667; MSL3; KLF13; ZNF669; GATA6; CREB3L1; CBX7; ZKSCAN1; ZSCAN18; ING4; RUNX1; HIVEP1; NFYC; NR4A3; TBX10; ZNF184; ZNF580; KDM4A; FOXI1; SOX18; RORA; ZNF446; ZKSCAN4; TRIM22; HTATIP2; EVX1; TULP3; ZNF358; SREBF2; INSR; FOXH1; BRF2; ATF6B; ZNF337; MYOD1; ZFPM2; SIX5; POU4F2; FOXO3; DCC; TCF15; SIX6; HNF4G; NKX2-5; TCF7; TBX1; ESRRB; ZNF350; ID2; REL; ZNF195; CEBPD; TBX5; FOSL2; ZNF529; ZFHX2; MAF; ZNF264; ZNF362; POU2F1; SOX3; ARID3B; MEIS1; UTF1; CARF; NFE2; POU2F3; TAL1; ZBTB39; CTCF; SKI; AFF2; SCAI; POLR3C; PIR; HIRA; TERF1; GLI2; ZNF74; ZNF768; BHLHE41; LMCD1; ZSCAN31; CRX; HOXD13; ZNF611; ZNF671; MAFG; RFX3; DACH1; FOXN3; ZNF215; TAF6L; NCOA3; ELF3; RYBP; ZNF155; DYRK1B; ZBTB3; HIC2; SMARCC2; PRDM14; HLX; HOXD1; THRA; IRF1; SRCAP; NCOA1; GCM1; SALL2; HOXD9; TAF1C; ZNF665; MED12; KLF4; ZBED1; PRDM12; MEF2D; NFATC1; ZNF124; STAT5A; ZXDC; ZNF266; NKX3-1; HOXA3; BRD4; BARX1; ZFHX3; BNC2; APBB1; HEY2; ZNF394; TOX; HNF4A; TCF4; ZNF589; HNF1A; ZNF770; VENTX; ZNF225; MYF5; VDR; BARX2; KLF1; ZNF682; ZNF257; ZNF516; ONECUT1; LPIN2; ZBTB44; DDIT3; TCF21; MAML3; RFX1; TEAD3; ZNF268; PRDM9; HIF3A; SETDB1; TSHZ2; ZNF423; CEBPE; KAT6A; SALL1; RING1; IKZF3; EMX1; ZNF331; TDP2; AEBP1; SKIL; SOX17; MXI1; ZIM2; ZNF652; HOXB13; TGIF1; NFATC3; MAFB; ZNF814; ZNF12; LIN28A; CREM; MAPK8IP1; JAK2; HOXC5; KLF15; MDM2; NR4A2; NKX2-2; HOXB2; TGIF2; ZNF467; ZNF532; TFEC; HOXD11; FOXA2; TRIM29; ZNF440; L3MBTL1; ANKRD1; KLF3; MAK; SRY; HDAC4; CERS4; RORC; NR1H2; FOXO1; TRIM16; LYL1; ASH2L; ZNF112; SMAD2; ZNF345; NR4A1; ZNF219; ZHX2; PKNOX2; NR0B1; JUP; ATF4; NFIC; YBX2; ZNF623; TP53; CEBPA; TP73; BACH2; NR1D2; MYCN; RFX5; FEZF2; ZNF85; TCEA2; PRDM1; BRD2; ELF5; ZNF536; SOX13; STAT1; CUX1; TLE2; WWP1; SOX2; KLF11; ATF3; ZNF93; MED13; SCAND1; RUNX3; PAX8; ID4; SATB2; SSBP3; RSF1; AES; BCL11B; DLX5; PBX1; ZIC3; ATN1; MYCL; IRF6; SOX10; TP63; KAT6B; NANOG; ERBB2; EMX2; IRF8; CBFA2T3; TRIB3; BCL11A; WT1; ERBB4; POU2AF1; STAT4; NFE2L3; NCOA2; SHOX2; ARID5B; IRF7; AR; HDAC9; NPAS2; BACH1; ZFP36L2; MECOM; VGLL4; XBP1; FLI1; JUND; TXNIP; MYB; CREB1; LEF1; TOX3; IFI16; THAP11; EHF; HLF; ID3; MEIS2; ARNT2; MNDA; PAX5; TFAP2C; TLE1; ESR1; BASP1; FOS
Down-regulation 119 FOSL1; CCNA2; MYC; MYCBP; PARP1; HMGA2; EGR1; TFDP1; RUVBL2; DR1; RUVBL1; HDAC2; NELFB; WHSC1; NUP62; TBP; SUB1; EZH2; DRAP1; UBE2I; CENPF; PMS1; PTTG1; TCERG1; SLC2A4RG; SMARCA5; BMI1; CBFB; BAZ1A; RHOA; PA2G4; HNRNPD; BRCA1; CBX3; CAPN15; RNF4; CALR; WDHD1; ZNF146; NR2F6; HOXA1; HES1; TRIM28; TEAD1; RBM14; PSMC3IP; HMG20B; HLTF; FOXD1; ETV1; PPRC1; BCLAF1; SSRP1; SMARCA1; BRPF1; CBX5; RBL1; HSF2; ASXL1; ING2; ADRB2; RBPMS; BAZ1B; GTF2IRD1; URI1; HIPK3; TAF9; APEX1; PITX1; NONO; SOX9; CNBP; RBBP7; NFIB; NPM1; RBBP8; ELK3; GTF2I; CEBPZ; BRIP1; RAN; SAP30; DLX2; HMGB2; EGR3; MTDH; MBD2; MAFF; MYBL1; NRIP1; FOXM1; RBBP4; BRD3; BLM; EED; SMAD5; ITGB3BP; SMARCA4; IRX5; EDF1; HMGB1; NAB1; TGFB1; DEK; ZBED2; SUV39H1; TBL1X; NR1H3; AHR; HMGA1; KLF9; SMAD3; SPEN; PBX3; MYBL2; CREB3L2; STAT3; HOXC6; PUF60