Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17425 Canertinib GSE70138 MCF10A Human 24h 0.12uM EID0020
Types Number Response transcription factors
Up-regulation 280 TSC22D3; PNRC1; NFKBIA; ZNF665; ZNF768; BTG1; VGLL4; ZMYM2; ING4; ZBTB44; ZNF611; TRIM29; AFF2; IRF6; CSDC2; BPTF; E2F5; CARF; ZNF44; ZKSCAN8; RFX5; HOXB3; SOX4; CALCOCO1; TRPS1; MTF1; NR5A1; TRIM16; TEAD3; ASCL3; RARB; ZNF345; CREG1; ZNF160; ZKSCAN4; FOXO4; ZNF91; ZKSCAN1; RING1; MXI1; ZNF264; SSBP3; HDAC5; ID2; MECP2; ADRB2; NR1H2; MYCL; TRIM22; PBXIP1; ZNF254; ZMIZ1; ATF3; ZNF224; KLF3; OSR2; KDM4A; GATA6; ZFHX3; ZNF34; ARHGAP35; FOSL2; CREBL2; CBX7; MZF1; MEIS2; ZNF711; AR; ZNF430; SPI1; ZNF467; WNT4; MDM2; RCOR3; ZNF250; REPIN1; SOX12; ZNF136; MEF2C; THRB; ZNF117; ESRRA; SMARCD2; CBFA2T3; LDB1; TP63; ZNF500; TSHZ2; ZNF652; JUP; ZNF536; REL; SP3; ZNF667; PBX1; CEBPD; BCL6; ATOH1; ZIM2; AES; ZSCAN31; HBP1; TCEB2; MEIS1; ZNF331; IRF3; PKNOX2; RORC; TCF7L2; TOX3; ZNF573; HMBOX1; ZNF24; MED13; SCAI; RARG; ZSCAN9; PCGF2; HIF3A; ZNF124; ZNF701; STAT2; FOXO3; ZNF629; FOSB; ERBB2; CHD8; DLX5; SIM1; ZNF358; ZNF3; CUX1; CIR1; SOX13; PHIP; SALL2; ZNF226; ZNF444; TGIF1; PEX14; CBX4; NFAT5; TFCP2L1; ZNF195; ZNF623; PDLIM1; NR1H3; ZBTB1; ZNF75D; ZNF688; LITAF; BCL11A; CEBPA; FOXF1; PAWR; ZNF14; TFEC; ZBTB20; ZNF587; PEX2; CHD4; ELF1; RSF1; ZNF12; DBP; ZNF426; ARID1A; CD3D; SOX3; EPAS1; CHD9; ERF; ZNF7; SMARCD3; NFIX; SUPT4H1; ZNF544; SP140; CERS4; ZNF516; SCAND1; NLK; BAZ2B; KAT2B; IRF9; MNDA; MITF; OLIG2; ZKSCAN7; SKI; FOXN3; ISL1; ZNF304; ZNF43; INSR; ZNF721; SRCAP; INSM1; ZNF112; HEY1; TRIM24; MED24; ZNF85; ASCL1; NFATC4; ZNF268; FOXF2; ZNF415; ZIC3; TCF7; ZBTB16; IRF2; HOXB5; ZNF468; SIX2; SNAI2; DDX17; SPIB; TXNIP; TCF25; TP53; HOXB2; FOXO1; ZNF83; TCF12; KDM5C; ATN1; ZNF350; PAX5; NCOA3; TCF7L1; ZNF93; TCF21; MAF; EHF; NCOR2; ZHX2; CERS6; ZIC1; ELF4; MED1; BRD2; CITED2; FOXA1; ELF3; PEG3; MKL2; CREB3L2; DAXX; TLE1; ID1; ZNF551; GRHL2; BNC2; SP110; PLAGL1; MECOM; ZMYND8; TCF4; WT1; NR4A2; FLNA; HOXB6; ARNT2; JUND; MYCN; GLI2; POU2AF1; MYRF; HMGN3; ID3; TSC22D1; EMX2; FOXG1; ARID5B; ESR1; TBX3; HMG20B; SSBP2; ZNF586
Down-regulation 76 CCNA2; FOSL1; HMGA2; BRCA1; EZH2; NRIP1; CDK2; SUV39H1; CENPF; NUP62; FOXM1; TFDP1; PTTG1; RUVBL1; DNAJC2; MYBL2; WHSC1; CHAF1B; PARP1; HNRNPD; CRY1; FHL2; DRAP1; GMNN; HMGB2; TEAD4; CCNE1; ING2; PSMC3IP; PPRC1; ILF2; PA2G4; TAF9; BMI1; RBM14; RAN; PSMC3; RNF4; BCLAF1; PREB; ELK3; EDF1; CBFB; ETV4; BLM; NFIB; DEK; HMGB1; NOC2L; EED; RBL1; RB1; CAMTA1; ZNF143; CEBPG; NPM1; XBP1; RUVBL2; DNMT3B; CTR9; SMAD3; CEBPZ; MYBL1; HMGA1; ZEB1; WWTR1; TRIM28; ARNTL2; EGR3; PURA; BHLHE41; EGR2; HOXC6; MYB; BASP1; KDM5D