Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17421 Canertinib GSE70138 MCF10A Human 24h 10uM EID0020
Types Number Response transcription factors
Up-regulation 381 TSC22D3; PNRC1; FOXO4; ZNF117; CALCOCO1; TRIM16; TCFL5; AFF2; NR1H2; IRF7; IRF9; CSDC2; ZNF91; ZKSCAN4; ZNF345; HDAC6; RFX5; ZNF423; NR5A1; NCOA2; ZNF362; ZNF768; ASCL3; ZBTB3; TBX6; ZNF611; ZFPM2; TLX1; SMAD6; CDX1; REL; SOX17; PBXIP1; ZNF688; JUP; ZIC4; ZFHX3; ZBTB44; VGLL4; HIVEP1; ZNF44; HDAC5; AR; NR3C2; TBX4; ING4; ESR2; MDM4; SOX18; NKX3-2; ZNF254; HIF3A; TAF1C; SP2; ATOH1; ZNF154; ARID5A; HOXB1; GCM1; ZNF132; ZNF184; CHD2; BARX1; KAT2B; THRB; THAP7; RORC; ZNF224; PPARA; ZKSCAN1; ZNF652; MZF1; MYCL; NFYC; THRA; ALX3; MAML3; POU6F1; TEAD3; MXI1; CARF; ZSCAN9; BTG1; ETV2; HNF4G; ZNF507; SPI1; RING1; SMARCC2; DYRK1B; CRX; ZFHX2; ELF4; PRDM9; FEZF2; TFEB; HBP1; ERBB4; ZNF93; ZNF467; SOX3; TBX5; ZNF665; SSX3; ZNF358; HOXB3; SALL2; MYF5; MEF2C; RARB; ZNF500; ZIC1; ZHX2; ZNF136; ZNF174; VGLL1; NEUROG1; RBBP5; NEUROG3; PKNOX2; IKZF3; WT1; ZNF43; TRIM29; CBX4; CBX7; PEX14; BHLHE41; RFX1; ZNF354A; ETV7; RBPJL; ZNF264; ZNF219; NR1I3; TRIM22; TSHZ2; ZNF74; ZNF124; ZNF274; MEIS2; PRDM12; CDX2; IFNB1; ZNF669; PROP1; CERS4; STAT2; CBFA2T3; MED13; LMX1B; WNT4; ZNF253; TP73; PHIP; VENTX; FOXH1; KLF3; SUPT7L; EVX1; ZNF671; MAK; HSF4; MECOM; ID2; SIX5; PHF1; ZNF14; SIX3; TULP1; CHD9; GBX1; FOXN3; FOSL2; YBX2; POU4F3; ZSCAN2; ZNF778; FOXI1; HOXA3; SSBP3; TCF7; MEIS1; SNAI1; ZNF195; RARG; ZNF430; PRDM1; TAF6L; ZNF257; ZBTB7B; HIVEP3; KLF13; KLF11; ZNF273; ZNF682; ZNF141; CBFA2T2; CEBPE; PRDM14; ZNF34; CEBPD; GBX2; MNDA; DLX4; RAX; MED12; CIR1; TCEA2; PLAG1; TBPL1; SKIL; LHX3; MECP2; IRF1; HINFP; SIX6; ZNF160; THAP10; CREBL2; ZSCAN31; ZNF771; TBX1; KDM4A; L3MBTL1; TOX; NFAT5; INSR; TFAP2A; SIM1; POU2AF1; ZIC3; EZH1; ZNF701; SIX2; ZNF223; TLE2; CDIP1; EHMT2; TLX3; ZNF12; TSG101; ZNF205; ATF3; HIPK1; ZNF140; ZNF85; HOXD1; PPP1R13L; SOX21; SOX13; NKX3-1; TCF15; TULP3; LYL1; KAT6B; PAX8; ZNF580; ZNF222; SP100; REPIN1; ZNF268; MSC; ZNF394; RYBP; ZNF426; TFEC; ZNF33B; SALL1; CREM; ZSCAN16; ZNF331; CREB3L1; RORA; NFE2L3; MEN1; SP110; ZNF444; SCAND1; IRF6; TBX2; SUPT4H1; JAK2; SRCAP; BCL11A; GTF2IRD1; ATN1; BACH1; STAT1; ETV6; GATA1; TCF4; NFATC4; BNC2; PIR; ZBTB43; FOXF1; CUX1; PRDM2; TERF1; ELF3; TP53; TERF2; GRHL2; PCGF1; RSF1; HOXB13; TAF7; TCF21; BAZ2B; TFAP2C; NR0B2; ZKSCAN7; ARID1A; CRYM; MYT1; ZBED2; ELF5; OVOL2; TP63; BCL6; ZNF606; PLAGL1; NCOA3; HOXB5; HIRA; EMX2; NFE2; SP140L; ZBTB20; FOSB; OSR2; IRF2; DLX5; SOX11; TAL1; ZNF217; TRIB3; TWIST1; FOXO3; TDP2; NPAS2; ZEB1; HIC2; ZNF350; ARID5B; RXRA; TFDP2; ISL1; MAFB; FLI1; DAXX; CUX2; DACH1; SSX1; ZBTB16; SHOX2; TCF7L1; FOXA2; ST18; LITAF; AES; SOX10; ARNT2; JUND; PBX1; NR0B1; GATA6; FOXF2; TXNIP; HTATIP2; TLE4; SNAI2; FOXC1; IFI16; KLF5; VPS72; CREB1; NR4A2; SOX2; HMG20B
Down-regulation 125 CCNA2; FOSL1; HMGA2; TFDP1; MYCBP; MYC; BRCA1; PARP1; TCERG1; HDAC2; ADRB2; RHOA; RUVBL1; EGR1; SUV39H1; CENPF; NRIP1; DNAJC2; HNRNPD; EZH2; FHL2; NUP62; PA2G4; RBBP7; BCLAF1; PSIP1; PTTG1; SFPQ; NEDD8; UBP1; HES1; C1QBP; RBM14; SMARCC1; RUVBL2; PPRC1; MYBL2; HMGB2; NPM1; CBFB; XRCC6; SSRP1; ATF1; TRIM28; RNF4; SUB1; ING2; ENO1; WDHD1; NFIB; PMS1; CHD1; DRAP1; BAZ1A; HMGB1; RFC1; YBX1; DR1; CAPN15; RNF138; NOC2L; HOXA1; ZNF146; UBE2I; ORC2; RB1; HOXC6; SF1; CNOT1; SMARCE1; HSF2; RBPMS; TFAM; DEK; CBX3; EGR3; RBBP4; MTF2; ILF2; TRRAP; RAN; CEBPZ; FLNA; AGO2; FOXM1; WHSC1; BHLHE40; AATF; BCL11B; EDF1; DNMT3B; HLTF; PRKDC; EGR4; HDAC1; PSMC3IP; URI1; ASCL1; ELF1; HSBP1; RNF14; SMARCA2; MTA1; TAF9B; YWHAB; AHR; MTDH; HOXB7; BMI1; ING3; NR2F2; PUF60; TBL1X; HIPK3; SOX9; HOXC10; FOXD1; SAP30; CALR; ELK3; EGR2; KLF10; TRIP6; PEG3; DMTF1