Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID17200 Canertinib GSE70138 MCF10A Human 24h 0.37uM EID0019
Types Number Response transcription factors
Up-regulation 225 TSC22D3; FOXO3; ZMIZ1; MEIS1; NFKBIA; FOSL2; ING4; CREG1; PBX1; TRIM22; PNRC1; PBXIP1; TRIM29; CALCOCO1; TLE1; NCOA3; SOX4; ZNF768; SRCAP; SREBF2; IRF6; JUP; ELF3; TP53; ZNF268; ZKSCAN4; CBX7; CEBPD; ZMYM2; ZNF358; ZNF629; BPTF; HDAC5; TP63; SUPT7L; FOXN3; ZFHX3; LDB1; ELF4; ESRRA; EP300; NFE2L2; BAZ2B; BCL6; ZNF345; TRPS1; HBP1; BTG1; ZNF112; ZSCAN9; RSF1; SALL2; SREBF1; HMBOX1; KDM4A; EZH1; WNT4; ZNF12; ZNF688; ID2; ARHGAP35; SOX12; CHD9; RING1; CSDC2; ZNF669; EHF; TSHZ2; NR5A1; ZMYND8; TCEB2; MED23; ZNF611; MECOM; MZF1; ZNF354A; VGLL1; TEAD3; SOX17; SOX3; ZNF331; ZBTB16; NFE2L1; ZHX2; ZNF665; ADRB2; ID3; NFIC; ZNF467; ZBTB7A; TRIM16; CIR1; PRDM2; NFATC4; LYL1; NCOR2; ZNF44; ZNF652; CERS4; IRF9; ZNF623; OVOL2; MKL1; ZSCAN31; ZNF33B; TFCP2L1; CUX1; TRIM24; ZSCAN32; TCF25; AES; DDX17; HEY1; ZNF606; EPAS1; ZNF415; ZNF573; ZNF667; MAF; CREBL2; GRHL2; MEIS2; ZNF544; ZNF91; E2F5; ZNF468; ZNF136; NCOA2; ZNF426; ZNF83; OSR2; AHR; ZSCAN16; CBX4; ZNF219; FOXO1; HIVEP1; RARG; CNOT2; ZNF93; ZNF532; MECP2; ZNF224; CBFA2T3; ZNF165; ERBB4; PDLIM1; THRA; MXI1; ZKSCAN1; RXRA; HIPK1; ZNF160; NFAT5; REPIN1; CDIP1; ZNF304; ZNF423; INSM1; ZKSCAN7; MED13; ZNF117; MYCL; NR4A2; ZNF350; ZNF430; DLX4; VGLL4; KLF5; ZSCAN18; RUNX1; NAB1; DLX5; ERBB2; SOX2; INSR; MYCN; ID1; TCF4; ZNF512B; TCF12; ZBTB20; TOB1; ZFPM2; NR1D2; BCL11A; NFATC1; REL; SSBP3; NR1H2; SMARCD2; STAT1; NEUROD1; CEBPA; PAWR; ATF3; ESR1; TFEC; JUN; ARNT2; FOSB; PEG3; LITAF; SNAI2; ZNF264; TSC22D1; MAFB; TOX; SCAND1; TXNIP; TBX3; HTATIP2; ZNF43; ZNF721; TFAP2C; TGIF1; ZIC1; GATA6; RFX5; ARID4B; FOXO4; SSBP2; GATA3; BASP1; FOS
Down-regulation 95 CCNA2; FOSL1; MYBL2; FOXM1; HMGA2; CENPF; CDK2; NUP62; SUV39H1; TCERG1; PTTG1; HMG20B; EGR1; HMGB2; FHL2; WDHD1; EZH2; PSMC3IP; CHAF1B; RBL1; NPM1; GMNN; ETV4; RNF138; RBM14; DRAP1; MYBL1; E2F1; RUVBL1; ITGB3BP; YEATS4; BATF3; WHSC1; BRCA1; DR1; PSMC3; DNMT1; HNRNPD; HMGB1; PA2G4; SAP30; SSRP1; TFAM; BLM; ALX1; TAF1A; EGR3; HOXC10; BCLAF1; CBFB; EGR2; WWTR1; BMI1; CCNE1; TEAD4; RAN; HOXB7; GATAD2A; HHEX; BRIP1; HLTF; BAZ1B; BAZ1A; EED; DNMT3B; CEBPG; XBP1; CRY1; ETS1; SMAD3; HOXC4; CBX5; SFPQ; ETV1; NR2F1; DEK; ILF2; CHD7; YWHAB; ING2; KLF6; TRIM28; FOXD1; POU4F1; HOXC6; KDM5D; IRF4; LEF1; PBX3; SUB1; AEBP1; BHLHE40; SATB2; PPARG; SATB1