Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID12301 Canertinib GSE70138 HME1 Human 3h 0.12uM EID0018
Types Number Response transcription factors
Up-regulation 69 THAP7; TAF5; E4F1; KLF3; TSC22D3; ZNF580; ZNF688; EN1; VDR; JUP; TCEA1; ZHX2; HOXA5; NR5A2; MEIS2; CERS4; NFKBIA; ZNF423; FOXM1; HHEX; ZNF232; BARX1; NFATC4; TWIST1; ZNF467; KLF11; FOXG1; HBP1; TULP3; PITX2; NR1H4; BNC2; SPDEF; SMAD1; ZNF512B; SCAND1; TCEA2; NANOG; FOXO1; ID2; TFAP2A; CEBPD; MXI1; PIR; NFE2L3; TFAP2C; TOB1; SOX11; ARNT2; PBX1; BCL11A; LIN28A; WT1; SOX17; MEOX2; MYBL1; TLE4; TRIB3; ZFPM2; THAP11; TEAD4; HOXB7; AEBP1; EMX2; MECOM; HMG20B; ESR1; ID1; POU2AF1
Down-regulation 48 MYC; HMGA2; NR4A1; EGR3; NR4A2; CHD1; ZBTB38; ATF1; HLTF; FOSB; TMF1; ZNF443; EGR1; SMARCA4; TSC22D2; HSBP1; SFPQ; NRIP1; SATB2; ING3; ZEB2; CTNNB1; ETS2; BAZ1A; ELK3; ZNF587; CHD7; FOXC1; CREB3L2; TFAM; TGFB1; SMARCA2; NFAT5; JUNB; AHR; SOX9; BAZ2B; LEF1; NCOA1; ZNF160; HMGN3; BHLHE40; ERG; TBX3; EGR2; TOX3; MSX1; TCFL5