Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID12066 Canertinib GSE70138 HME1 Human 3h 3.33uM EID0017
Types Number Response transcription factors
Up-regulation 22 TSC22D3; NFIL3; EZH1; XBP1; TOX; CARHSP1; ZBTB20; TCEA1; HOXD11; TRIB3; HMGB2; SATB1; TAL1; PIR; NR2F2; HOXC10; HOXB7; CITED2; EMX2; WT1; TOB1; ARNT2
Down-regulation 29 MYC; HMGA2; FOSL1; JUN; ETS1; NRIP1; URI1; EGR1; KLF6; ABL1; CTBP1; ADRB2; ERG; EGR3; HLX; SMAD7; SATB2; NR2F6; SIX1; AHR; WWTR1; SMAD3; ELK3; TBX3; IRX5; SOX9; ASCL1; TSC22D1; KDM5D