Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID11836 Canertinib GSE70138 HME1 Human 3h 0.37uM EID0016
Types Number Response transcription factors
Up-regulation 56 MYBL2; TSC22D3; NFE2L2; OVOL2; ZNF189; DMRT1; PQBP1; ID2; PSMC3; TFAP2C; POLR3C; NCOA3; FOXN3; TCF3; ARID5B; ZNF354A; RNF138; NFIL3; NCOA4; WWC1; NFE2L1; E2F8; STAT1; MYCN; ZSCAN31; XBP1; SREBF1; MYRF; NANOG; JUP; ID3; ELF5; FLI1; TLE4; SAP30; ZBTB16; MYB; SIAH2; CUX2; MYBL1; CBFA2T3; TRIB3; EGR2; HOXB7; TRIM29; ST18; OSR2; NKX2-2; BHLHE41; MNDA; TRIM22; KAT6B; ZFP36L2; PEG3; ID1; MAFB
Down-regulation 47 FOSL1; MYC; JUN; TCERG1; JUNB; UBE2I; ABL1; FOXF1; FOSB; HMGA2; ALX1; FOXD1; CHD3; ESRRG; MYT1L; BHLHE40; BCL3; SERTAD2; RORA; CRY1; NR4A1; EGR3; LPIN2; MECOM; MED1; SMARCD3; CREB3L1; NR4A2; LOXL2; SHOX2; LEF1; NR2F1; TSC22D2; PAX5; SMARCA1; ELK3; HEY1; BTG1; ZNF91; HMGN3; ZBTB18; SUB1; ZBTB20; KDM5D; ZFP36L1; ZIC1; IKZF1