Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID11835 Canertinib GSE70138 HME1 Human 3h 1.11uM EID0016
Types Number Response transcription factors
Up-regulation 69 NR1H2; TSC22D3; MEF2C; TFDP2; CBX7; ID2; SOHLH2; CEBPZ; TEAD3; EMX2; JUP; SIAH2; SMAD6; NCOA3; NELFB; PPARG; ST18; BRD7; ZSCAN31; PAWR; SUPT3H; RYBP; TRIB3; KLF5; SALL2; FOXF1; CEBPG; DDIT3; ERBB4; KLF11; ZFPM2; NFIL3; SUPT4H1; TLE4; MTF2; TFAP2C; KLF4; ID3; TFAP2A; ID1; YAP1; TCF21; PAX6; FOXA1; BNC2; MYRF; ZNF264; TAL1; CREB1; ATF4; ARNT2; RBPMS; ZSCAN18; NR4A2; ESR1; MEIS2; HIRA; ZHX2; HHEX; TGIF1; THAP11; AEBP1; IRF8; ZFP36L1; HTATIP2; ATF3; TCF4; HOXC6; HMG20B
Down-regulation 33 MYC; FOSL1; HMGA2; ADRB2; CRY1; CHD7; ZMIZ1; PFDN5; NFIC; BHLHE41; CBFB; BHLHE40; RREB1; JARID2; SIX2; BAZ1A; HNRNPD; TRIM32; MSX1; SMARCD3; EGR3; KLF10; SMAD7; ASCL1; PSIP1; FOXC1; ELK3; CREG1; CITED1; STAT4; TRIM22; KDM5D; TCFL5