Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID11382 Canertinib GSE70138 HME1 Human 24h 0.37uM EID0014
Types Number Response transcription factors
Up-regulation 105 NFATC4; BTG1; TSC22D3; MAK; MYCL; KAT2B; MAF; TP53; BCL11A; HDAC5; BAZ2B; BACH2; PRDM2; ZSCAN31; RLF; GLI3; PNRC1; CREG1; CDYL; EN2; ZNF536; NKX2-1; NFKBIA; AR; TRAK1; FOXN3; NFIL3; BCOR; ZNF248; OSR2; IRF1; HOXA5; CDX1; ZFHX4; TRIM16; STAT3; ZNF44; PAWR; LITAF; ZNF219; ZNF274; PPARG; CTBP2; ING4; KLF4; PRMT2; EDF1; INSM1; DACH1; ZNF580; ZEB2; YBX1; CREBL2; KLF11; INSR; STAT1; ATF3; DLX2; FOSB; SHOX2; JUNB; MXI1; NCOA1; RYBP; NR4A1; ZSCAN18; CHD7; HBP1; IRF6; ERBB2; FOXJ3; PAX6; SPIB; BCL6; SATB2; MEIS1; ZNF331; CREB1; TLE1; TSC22D2; ZNF573; PLAGL1; ZMIZ1; TOX3; MTA1; MEOX2; CEBPD; ZNF91; TCF7L1; MTF2; TLE4; ZBTB38; PSIP1; ELF3; LOXL2; THAP11; PBX1; GATA6; EMX2; ZBTB18; PAX5; ETS2; SOX11; MYB; SSBP2
Down-regulation 39 EGR1; HMGA2; SETD3; ARNTL2; BLZF1; TGFB1; ILF2; EGR4; ETV4; ETV5; BHLHE40; SMAD2; FOXD1; HMGA1; HOXC10; XBP1; SOX9; GATAD2A; ZNF593; HIRA; DNAJC2; TOB1; CBFB; PRRX1; BATF3; CD3D; NKX2-2; JUND; ZNF22; MYBL1; TSC22D1; TRPS1; KLF2; MSX1; NR2F6; MAFB; ID1; TBX2; ZNF586