Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID11381 Canertinib GSE70138 HME1 Human 24h 1.11uM EID0014
Types Number Response transcription factors
Up-regulation 106 PCBD1; TP53; KDM5A; MEF2C; FOSB; CNOT2; CREG1; HDAC6; TSC22D3; ZSCAN31; MZF1; MXI1; TCEA2; MEIS2; NFKBIA; NFIX; WNT4; EHMT2; BRD2; BCL6; SUPT3H; TRIM16; CALCOCO1; HOXA5; HLF; ZIC1; SHOX2; ZFHX3; JUN; NR1H4; SOX2; BCL11A; NFKB2; FOXO3; ATF3; PITX1; TBL1X; IRF9; ZNF444; MAFB; KAT6B; ZNF768; AIP; TULP3; BTG1; TEAD3; OSR2; ZNF219; CDIP1; CBX7; HHEX; SIX3; PAX6; MTA1; JUP; REL; CERS4; ZHX2; AHR; PFDN5; ING4; PBX1; TCEB2; NKX2-1; ELF1; PIR; TLE2; AES; NFE2; ERBB2; DDX17; CEBPD; TP63; HOXC4; CEBPZ; YAP1; VGLL4; KLF4; NKX3-1; DLX2; ZMIZ1; MITF; CBFA2T3; ESR1; FLNA; CUX1; TLE1; FOXF1; SMAD1; SCAND1; ZNF423; WWTR1; MEIS1; RBPMS; HMG20B; EMX2; TCF4; SOX9; PEG3; BACH2; DLX5; FOXG1; MECOM; ID1; ZFP36L1; SOX11
Down-regulation 50 TCERG1; HMGA2; PUF60; HMGB2; CENPF; RBM14; EGR1; ETV1; SUV39H1; AGO2; ELK3; HES1; ING2; CCNA2; SMARCA5; NRIP1; TAF1A; RCOR1; SUB1; PTTG1; DNAJC2; RAN; HSBP1; ZNF281; ZBTB11; NFE2L1; BHLHE40; RNF138; ARNTL2; XBP1; RAD21; OLIG2; NKX2-2; SFPQ; ZNF22; RNF4; SMAD7; SAP30; ZBED2; MNAT1; MYBL1; MAGED1; BHLHE41; TOB1; TGFB1; KDM5D; FOXD1; MYB; TOX3; TXNIP