Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID10018 Gsk-461364 GSE70138 HA1E Human 24h 0.04uM EID0077
Types Number Response transcription factors
Up-regulation 59 PPARG; ADRB2; NR1I2; ZBTB7A; NR3C2; MTDH; NCOR2; NFATC3; CARM1; CRK; DNAJC2; YWHAB; HOXA1; KDM2A; TCERG1; CCDC59; PBX2; KAT6B; CTR9; COPS5; ARID4A; ZNF131; SOX10; HOXD1; MTA1; BMI1; IRF4; SMAD6; ZMYND8; MYCN; MEOX1; HOXA5; NR2F6; SMAD7; GATAD2A; SMAD3; TBPL1; HOXB7; NFAT5; HLX; MECOM; FOS; HEY1; ZEB1; SNAI2; SATB2; ZNF217; CHD7; FOXD1; MSX1; ZNF589; FLNA; LEF1; NR4A2; ID3; TOX3; KLF5; ID1; SOX9
Down-regulation 60 NFKBIA; SHOX2; JUN; TAF1D; ACTL6A; MYC; LOXL2; PAWR; HBP1; SMAD1; TOX; JUND; IRF9; ISL1; ELF3; CALCOCO1; RORA; ZBED1; CTBP2; SOX4; PAX5; CDK2; ASCL1; ATF3; KLF7; AR; TSC22D1; ZBTB16; NKX2-1; PBX3; CREB1; NR4A1; FOXG1; ZNF232; YEATS4; ZFP36L2; MEIS1; PFDN5; FOXF1; ZNF331; BASP1; TXNIP; TRIB3; KLF10; CALR; TFAP2C; VPS72; EMX2; OSR2; BTG1; PITX1; SPDEF; FOXJ3; TLE4; KDM5D; STAT1; SSBP2; INSR; MYBL1; ESR1