Transcriptional response

Response ID Perturbagen Data accession Cell Source Species Duration Concentration Expression ID
RID08592 Canertinib GSE70138 HA1E Human 24h 3.33uM EID0012
Types Number Response transcription factors
Up-regulation 71 ZNF274; KLF5; AEBP1; NR4A1; TFAP2C; PIR; AHR; CBFA2T2; SP2; TCF20; ZNF721; TXNIP; NPAS2; ZBED1; ELF3; HTATIP2; NR4A2; EHF; SOX10; CNOT6; ZNF83; L3MBTL1; ID4; TAF9B; TDP2; POU2F1; MYCL; NR4A3; KDM5D; EYA1; CBX5; YBX3; ETS2; UBE2B; HMGB1; KLF6; ZNF711; GRHL2; ZMYND11; ZNF432; ID1; SMARCE1; HES1; PHIP; ZNF160; KLF11; IFI16; TRIM29; ZNF43; ZNF611; KLF4; E2F3; FOXA1; RUNX1; TP53; PPARG; MITF; ATF3; SATB1; ID3; ZNF331; TLE4; ZBTB20; MECOM; OSR2; KLF9; TOX3; DACH1; TBX3; NFATC3; LEF1
Down-regulation 52 HOXA5; COPS5; SMARCA1; ZNF281; RORA; ZNF146; ZZZ3; NFIC; ZNF148; ZBTB18; CEBPG; ZNF410; ZIC1; PRRX1; SSBP3; MTDH; COPS2; ZBTB11; IKBKAP; SMAD7; ZNF654; GFI1; MXI1; NR2F1; ZNF12; MSX1; GATA6; RBBP8; CITED2; BRD2; SP3; WT1; CALR; KLF7; ZBTB16; KLF2; CENPF; SMAD1; HOXB6; FOXO1; SHOX2; TGFB1I1; TAF10; IRF4; MYBL1; PLAGL1; SOX17; CEBPZ; HOXB7; PEG3; GATA2; ADRB2