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Database
Overview
Perturbagen
Expression Profiles
Transcriptional Responses
Download
Documentation
Contact
Home
Webtool
Database
Overview
Perturbagen
Expression Profiles
Transcriptional Responses
Download
Documentation
Contact
Targets of perturbagens
Perturbagen ID : CID56885
Perturbagen : 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide; Alpha-(4-methyl-1-piperazinyl)-3'-((4-(3-pyridyl)-2-pyrimidinyl)amino)-p-toluidide; Apo-imatinib; Gleevec; Imatinib; Imatinib mesylate; Imatinib methansulfonate; Imatinibum; Mylan-imatinib; Nat-imatinib; Pms-imatinib; Ran-imatinib; Sti 571; Teva-imatinib
Target
Effect
Reference
ABCB11
-1
STITCH
ABCG2
-1
CLUE; STITCH
ABL1
-1
DrugBank; CLUE; STITCH
ABL2
-1
STITCH
AKT1
-1
STITCH
BCL2L1
-1
STITCH
BCR
-1
CLUE; STITCH
BCR/ABL fusion
-1
DrugBank; STITCH
CSF1R
-1
DrugBank; CLUE; STITCH
CYP2C19
-1
CLUE; STITCH
CYP2C8
-1
CLUE; STITCH
CYP3A4
-1
STITCH
CYP3A5
-1
CLUE; STITCH
CYP3A7
-1
STITCH
DDR1
-1
DrugBank; CLUE; STITCH
DDR2
-1
STITCH
FGFR1
-1
STITCH
FGFR2
-1
STITCH
FGFR3
-1
STITCH
FGFR4
-1
STITCH
FGFRL1
-1
STITCH
FGR
-1
STITCH
FLT1
-1
STITCH
FLT3
-1
STITCH
FLT4
-1
STITCH
FYN
-1
STITCH
KDR
-1
STITCH
KIT
-1
CLUE; STITCH; DrugBank
LCK
-1
STITCH
MCL1
-1
STITCH
NQO2
-1
STITCH
NTRK1
-1
DrugBank; CLUE; STITCH
PDGFRA
-1
DrugBank; CLUE; STITCH
PDGFRB
-1
DrugBank; CLUE; STITCH
PDGFRL
-1
STITCH
RAF1
-1
STITCH
RET
-1
DrugBank; CLUE; STITCH
SRC
-1
STITCH
STYK1
-1
STITCH
SYK
-1
STITCH
TEK
-1
STITCH
TIE1
-1
STITCH
YES1
-1
STITCH
ABCB1
1
STITCH
BCL2L11
1
STITCH
CASP3
1
STITCH
AXL
2
STITCH
BIRC5
2
STITCH
BLK
2
STITCH
BMX
2
STITCH
BTK
2
STITCH
CA14
2
STITCH
CA2
2
STITCH
CA6
2
STITCH
CA7
2
STITCH
CA9
2
STITCH
CDC42BPB
2
STITCH
CRKL
2
STITCH
CSK
2
STITCH
CXCL8
2
STITCH
DOK1
2
STITCH
DSTYK
2
STITCH
EPHA1
2
STITCH
EPHA10
2
STITCH
EPHA2
2
STITCH
EPHA3
2
STITCH
EPHA4
2
STITCH
EPHA5
2
STITCH
EPHA6
2
STITCH
EPHA7
2
STITCH
EPHA8
2
STITCH
EPHB1
2
STITCH
EPHB2
2
STITCH
EPHB3
2
STITCH
EPHB4
2
STITCH
ERN1
2
STITCH
ERN2
2
STITCH
ETV6
2
STITCH
FIP1L1
2
STITCH
GSK3A
2
STITCH
GSK3B
2
STITCH
HCK
2
STITCH
HUNK
2
STITCH
IGF1R
2
STITCH
INSR
2
STITCH
INSRR
2
STITCH
IRAK1
2
STITCH
IRAK2
2
STITCH
IRAK3
2
STITCH
IRAK4
2
STITCH
ITK
2
STITCH
JAK1
2
STITCH
JAK2
2
STITCH
JAK3
2
STITCH
LIMK1
2
STITCH
LIMK2
2
STITCH
LYN
2
STITCH
MAP3K10
2
STITCH
MAP3K11
2
STITCH
MAP3K20
2
STITCH
MAP3K21
2
STITCH
MAP3K7
2
STITCH
MAP3K9
2
STITCH
MAPK1
2
STITCH
MAPK14
2
STITCH
MAPK3
2
STITCH
MATK
2
STITCH
MELK
2
STITCH
MERTK
2
STITCH
MET
2
STITCH
MLKL
2
STITCH
MOS
2
STITCH
MUSK
2
STITCH
NFKBIA
2
STITCH
NIM1K
2
STITCH
NUP214
2
STITCH
PASK
2
STITCH
PBK
2
STITCH
PIM1
2
STITCH
PIM2
2
STITCH
PIM3
2
STITCH
PKDCC
2
STITCH
PTK6
2
STITCH
PTK7
2
STITCH
RELA
2
STITCH
RIPK1
2
STITCH
RIPK2
2
STITCH
RIPK3
2
STITCH
RIPK4
2
STITCH
ROR1
2
STITCH
SLC47A1
2
STITCH
SOX17
2
STITCH
SRMS
2
STITCH
STAT5A
2
STITCH
STK11
2
STITCH
STK40
2
STITCH
TBXAS1
2
STITCH
TEC
2
STITCH
TESK1
2
STITCH
TESK2
2
STITCH
TRIB1
2
STITCH
TRIB2
2
STITCH
TRIB3
2
STITCH
TSSK1B
2
STITCH
TSSK2
2
STITCH
TSSK3
2
STITCH
TSSK4
2
STITCH
TXK
2
STITCH
TYK2
2
STITCH
TYRO3
2
STITCH
VEGFA
2
STITCH
ZAP70
2
STITCH