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Database
Overview
Perturbagen
Expression Profiles
Transcriptional Responses
Download
Documentation
Contact
Home
Webtool
Database
Overview
Perturbagen
Expression Profiles
Transcriptional Responses
Download
Documentation
Contact
Targets of perturbagens
Perturbagen ID : CID54528
Perturbagen : Caprelsa; N-(4-bromo-2-fluorophenyl)-6-methoxy-7-((1-methyl-4-piperidinyl)methoxy)-4-quinazolinamine; N-(4-bromo-2-fluorophenyl)-6-methoxy-7-((1-methylpiperidin-4-yl)methoxy)quinazolin-4-amine; Vandetanib
Target
Effect
Reference
ABL1
-1
STITCH
ABL2
-1
STITCH
AXL
-1
STITCH
BLK
-1
STITCH
BTK
-1
STITCH
EGFR
-1
DrugBank; CLUE; STITCH
EPHA1
-1
CLUE; STITCH
EPHA10
-1
CLUE
EPHA2
-1
CLUE; STITCH
EPHA3
-1
CLUE
EPHA4
-1
CLUE; STITCH
EPHA5
-1
CLUE; STITCH
EPHA6
-1
CLUE; STITCH
EPHA7
-1
CLUE; STITCH
EPHA8
-1
CLUE; STITCH
EPHB1
-1
CLUE; STITCH
EPHB2
-1
CLUE; STITCH
EPHB3
-1
CLUE
EPHB4
-1
CLUE; STITCH
EPHB6
-1
CLUE
ERBB2
-1
CLUE
ERBB3
-1
CLUE; STITCH
ERBB4
-1
CLUE; STITCH
FGFR1
-1
STITCH
FGFR2
-1
STITCH
FGFR3
-1
STITCH
FGR
-1
STITCH
FLT1
-1
CLUE; STITCH
FLT3
-1
STITCH
FLT4
-1
CLUE; STITCH
FYN
-1
STITCH
HCK
-1
STITCH
IRAK4
-1
STITCH
KDR
-1
CLUE; STITCH
LCK
-1
STITCH
MAP4K5
-1
STITCH
MERTK
-1
STITCH
MKNK1
-1
STITCH
PDGFRA
-1
STITCH
PTK6
-1
DrugBank; CLUE; STITCH
RET
-1
CLUE; STITCH; DrugBank
RIPK2
-1
STITCH
SIK2
-1
STITCH
SRC
-1
CLUE; STITCH
STK10
-1
STITCH
TEK
-1
DrugBank; CLUE; STITCH
TYRO3
-1
STITCH
VEGFA
-1
DrugBank; CLUE; STITCH
YES1
-1
STITCH
ACVR1
2
STITCH
BMPR1B
2
STITCH
DDR1
2
STITCH
GAK
2
STITCH
KIT
2
STITCH
MAP2K5
2
STITCH
PDGFRB
2
STITCH
RPS6KA6
2
STITCH
SLK
2
STITCH
STK35
2
STITCH